Mon. Jul 28th, 2025

ACY-1215

ACY-1215Band: www.medchemexpress.comAn orally bioavailable HDAC6-selective inhibitor against HDAC4, HDAC5, HDAC7, HDAC9, HDAC11, Sirtuin1, and Sirtuin2CAS No:1316214-52-4 Chemical Name:Rocilinostat  VX-767 Molecular Formula C24H27N5O3 Molecular Weight 433.5 CAS Numbers 1316214-52-4 Storage Condition…

4SC-202

4SC-202Band: www.medchemexpress.comAn orally bioavailable benzamide and inhibitor of human class I histone deacetylases (HDACs) isoenzymes 1, 2 and 3, with potential antineoplastic activity. CAS No:1186222-89-8 AMG 234 Molecular Formula C30H29N5O6S2 Molecular…

(+)-JQ1

(+)-JQ1Band: www.medchemexpress.comA potent, high affinity, selective BET bromodomain inhibitorCAS No:1268524-70-4 Reparixin Molecular Formula C23H25ClN4O2S Molecular Weight 456.99 CAS Numbers 1268524-70-4 Storage Condition 0°C (short term), -20°C (long term), desiccated Solubility…

BCI-121

BCI-121Band: www.medchemexpress.comNovel SMYD3 inhibitor, impairing cancer cell growthCAS No: 432529-82-3   Chemical Name: 4-(Aminocarbonyl)-N-(4-bromophenyl)-1-piperidineacetamide LY2109763 References PubMed ID::http://www.ncbi.nlm.nih.gov/pubmed/18502893

AT-7519

AT-7519Band: www.medchemexpress.comA potent inhibitor of several CDK family membersCAS No:902135-91-5 Pexidartinib Molecular Formula C16H17Cl2N5O2.HCl Molecular Weight 418.71 CAS Numbers 902135-91-5 Storage Condition 0°C (short term), -20°C (long term), desiccated Solubility…

AGI-6780

AGI-6780Band: www.medchemexpress.comPotent and selective inhibitor of the tumor-associated mutant IDH2/R140QCAS No:1432660-47-3 Chemical Name: AGI6780; QCR-283; 1--3-urea Asunaprevir Molecular Formula C21H18F3N3O3S2 Molecular Weight 481.51 CAS Numbers 1432660-47-3 Storage Condition 0°C (short term),…

AEM1

AEM1Band: www.medchemexpress.comNovel inhibitor of deregulated NRF2 transcriptional activity in cancer, broadly decreasing the expression of NRF2 controlled genes, sensitizing A549 cells to various chemotherapeutic agents, and inhibiting the growth of…

(-)-SW203668 Hydrochloride

(-)-SW203668 HydrochlorideBand: www.medchemexpress.comMore potent enantiomer of SW203668 (AOB9773), a novel tumor-specific inhibitor of stearoyl CoA desaturase (SCD)CAS No: 1673556-44-9 and 1673558-51-4 (Free Base)   Chemical Name: R(-)-4-(Amino(phenyl)methyl)-N-(6-methoxybenzothiazol-2-)benzamide Hydrocloride AZD9498 Molecular Formula C22H20ClN3O2S…

Camalexin

CamalexinBand: www.medchemexpress.comApoptosis inducer of T-leukemia Jurkat cells; Antimicrobial secondary metabolite in plant immune system BQ-790 (sodium salt) Molecular Formula C11H8N2S Molecular Weight 200.26 CAS Numbers 135531-86-1 Storage Condition 0°C (short…

Birinapant

BirinapantBand: www.medchemexpress.comAn orally bioavailable, synthetic bivalent small molecule peptido mimetic of second mitochondrial-derived activator of caspases (SMAC) and inhibitor of IAP (Inhibitor of Apoptosis Protein) family proteinsCAS No:1260251-31-7 Chemical Name:TL32711…