Sun. Jun 1st, 2025

JTE-607 dihydrochloride

JTE-607 dihydrochlorideBand: www.medchemexpress.comCytokine release inhibitor, inhibiting production of IL-1ß, IL-8, IL-6, IL-10 and TNFalphaCAS No: 188791-09-5   Chemical Name: N-benzoyl]-L-phenylalanine ethyl ester dihydrochloride BI 2537 Molecular Formula C25H31Cl2N3O5 2HCl Molecular Weight 597.36…

GW788388

GW788388Band: www.medchemexpress.comPotent and selective inhibitor of TGF-beta type I receptor CAS No:452342-67-5 Chemical Name: 4-{4--pyridin-2-yl}-N-(tetrahydro-2H-pyran-4-yl)benzamide ACY-1216 Molecular Formula C₂₅H₂₃N₅O₂ Molecular Weight 425.48 CAS Numbers 452342-67-5 Storage Condition 0°C (short term), -20°C…

EVP4593 (CAY10470)

EVP4593 (CAY10470)Band: www.medchemexpress.comPotent inhibitor of NF-κB activation and TNFα production CAS No: 545380-34-5   Chemical Name: QNZ; N4-​-​4,​6-​quinazolinediamine; CAY10470 Ko 144 Molecular Formula C22H20N4O Molecular Weight 356.42 CAS Numbers 545380-34-5 Storage Condition…

Takeda-6d

Takeda-6dBand: www.medchemexpress.comPotent inhibitory activity in both B-RAF and VEGFR2CAS No:1125632-93-0 Enasidenib Molecular Formula C27H19ClFN5O3S Molecular Weight 547.99 CAS Numbers 1125632-93-0 Storage Condition 0°C (short term), -20°C (long term), desiccated Solubility…

PF-04979064

PF-04979064Band: www.medchemexpress.comA potent and selective PI3K/mTOR dual kinase inhibitorCAS No:1220699-06-8 Tofacitinib (citrate) Molecular Formula C24H26N6O3 Molecular Weight 446.5 CAS Numbers 1220699-06-8 Storage Condition 0°C (short term), -20°C (long term), desiccated…

BI-69A11

BI-69A11Band: www.medchemexpress.comATP competitive, dual inhibitor of AKT and NFkB pathwayCAS No: 1233322-09-2   Chemical Name: (E)-3-(3-(1H-benzoimidazol-2-yl) acryloyl)-6-chloro-4-phenylquinolin-2(1H)-one Quizartinib Molecular Formula C25H16ClN3O2 Molecular Weight 425.87 CAS Numbers 1233322-09-2 Storage Condition Refrigerator (4 °C)…

ML061 ( Myricetin)

ML061 ( Myricetin)Band: www.medchemexpress.comInhibitor of DNA Polymerase III Holoenzyme System, PrimaseCAS No:  529-44-2 Ganetespib Molecular Formula C15H10O8 Molecular Weight 318.24 CAS Numbers 529-44-2 Storage Condition 0°C (short term), -20°C (long…

GW-9662

GW-9662Band: www.medchemexpress.comIrreversible PPAR-gamma antagonist CAS No:22978-25-2 Chemical Name: 2-Chloro-5-nitro-N-phenylbenzamide SB-431543 Molecular Formula C₁₃H₉ClN₂O₃ Molecular Weight 276.68 CAS Numbers 22978-25-2 Storage Condition 0°C (short term), -20°C (long term), desiccated Solubility DMSO Purity…

Darglitazone Sodium

Darglitazone SodiumBand: www.medchemexpress.comNovel agonist of peroxisome proliferator-activated receptor-gamma (PPAR-gamma)CAS No: 149904-87-0 (sodium free: 141200-24-0) Chemical Name: CP-86325-2; 5-phenyl]methyl]-1,3-thiazolidine-2,4-dione sodium salt GSK-690694 Molecular Formula C23H19N2NaO4S Molecular Weight 442.46 CAS Numbers 149904-87-0…

BSI-201

BSI-201Band: www.medchemexpress.comA selective, irreversible and orally bioavailable inhibitor of PARP1CAS No:160003-66-7 Chemical Name:Iniparib CTEP Molecular Formula C7H5IN2O3 Molecular Weight 292.03 CAS Numbers 160003-66-7 Storage Condition 0°C (short term), -20°C (long…