Mon. Jul 7th, 2025

AR420626

AR420626Band: www.medchemexpress.comNovel FFA3 selective agonistCAS No: 1798310-55-0 Chemical Name: N-(2,5-Dichlorophenyl)-4-(furan-2-yl)-2-methyl-5-oxo-1,4,5,6,7,8-hexahydro-quinoline-3-carboxamide PF-04447946 Molecular Formula C21H18Cl2N2O3 Molecular Weight 417.29 CAS Numbers 1798310-55-0 Storage Condition 0°C (short term), -20°C (long term), desiccated Solubility DMSO Purity…

Ambrisentan

AmbrisentanBand: www.medchemexpress.comSelective endothelin type-A (ETA) receptor antagonist CAS No: 177036-94-1 Chemical Name: Letairis; LU-208075; (2S)-2-(4,6-Dimethylpyrimidin-2-yl)oxy-3-methoxy-3,3-diphenylpropanoic acid PF-04418951 Molecular Formula C22H22N2O4 Molecular Weight 378.42 CAS Numbers 177036-94-1 Storage Condition 0°C (short term),…

AF64394

AF64394Band: www.medchemexpress.comNovel selective GPR3 Inverse Agonist, the first small molecule inhibitor of GPR3 receptor function GM6004 Molecular Formula C21H20ClN5O Molecular Weight 393.87 CAS Numbers 1637300-25-4 Storage Condition 0°C (short term),…

AdipoRon

AdipoRonBand: www.medchemexpress.comNovel agonist of adiponectin receptors AdipoR1 and AdipoR2 CAS No: 924416-43-3   Chemical Name: 2-(4-Benzoyl-phenoxy)-N-(1-benzyl-piperidin-4-yl)-acetamide GSK2606417 Molecular Formula C27H28N2O3 Molecular Weight 418.5 CAS Numbers 924416-43-3 Storage Condition 0°C (short term), -20°C…

AC-264613

AC-264613Band: www.medchemexpress.comThe first agonist of the G-protein-coupled receptor (GPCR) protease activated receptor 2 (PAR2) CAS No: 1051487-82-1   Chemical Name: AC264613; (3R,​4S)​-​rel-2-​Oxo-​4-​phenyl-​3-​pyrrolidinecarboxyli​c acid 2-​​hydrazide EW-7200 Molecular Formula C19H18BrN3O2 Molecular Weight 400.27 CAS Numbers…

TRAM 34

TRAM 34Band: www.medchemexpress.comPotent inhibitor of the intermediate-conductance Ca2+-activated K+ channel, blocking Kv1.3, Kv1.4, Kv7.2+Kv7.3 and Nav1.4 Avibactam (sodium) Molecular Formula C22H17ClN2 Molecular Weight 344.84 CAS Numbers 289905-88-0 Storage Condition 0°C…

RY796

RY796Band: www.medchemexpress.comNovel and selective Kv2 channel inhibitor  CAS No: 1393441-53-6   Chemical Name: 2-(Dimethylamino)-5--N--benzamide Senicapoc Molecular Formula C21H27N3O2 Molecular Weight 353.46 CAS Numbers 1393441-53-6 Storage Condition 0°C (short term), -20°C (long term),…

RY785

RY785Band: www.medchemexpress.comNovel and selective Kv2 channel inhibitor  CAS No: 1393748-80-5   Chemical Name: 3-Methoxy-alpha-methyl-N--benzenepropanamide XMD8-95 Molecular Formula C21H20N4O2S Molecular Weight 392.47 CAS Numbers 1393748-80-5 Storage Condition 0°C (short term), -20°C (long term),…

PAP-1

PAP-1Band: www.medchemexpress.comSelective inhibitor of Kv1.3, voltage-gated K+ channel CAS No:870653-45-5 Chemical Name: 5-​(4-​Phenoxybutoxy)​psoralen LY3023417 Molecular Formula C₂₁H₁₈O₅ Molecular Weight 350.36 CAS Numbers 870653-45-5 Storage Condition 0°C (short term), -20°C (long term),…

NS11021

NS11021Band: www.medchemexpress.comPotent and specific activator of Ca2+ activated big-conductance K+ channelsCAS No: 956014-19-0 Chemical Name: 1-(3,5-Bis-trifluoromethyl-phenyl)-3--thiourea Elacridar Molecular Formula C16H9BrF6N6S Molecular Weight 511.24 CAS Numbers 956014-19-0 Storage Condition 0°C (short term), -20°C…