Wed. Jul 16th, 2025

PJ34 Hydrochloride

PJ34 HydrochlorideBand: www.medchemexpress.comPotent inhibitor of poly(ADP-ribose) polymerase (PARP) CAS No:344458-15-7 Chemical Name: N-(5,6-Dihydro-6-oxo-2-phenanthridi​nyl)-2-acetamide hydrochloride AZD-9295 Molecular Formula C17H17N3O2.HCl Molecular Weight 331.8 CAS Numbers 344458-15-7 Storage Condition - 4C Solubility 100 mM in…

MK-4827

MK-4827Band: www.medchemexpress.comAn inhibitor of PARP 1 and 2CAS No:1038915-60-4, 1038915-64-8 Chemical Name: Niraparib  MK-1779 Molecular Formula C19H20N4O HCl Molecular Weight 356.85 CAS Numbers 1038915-60-4 Storage Condition 0°C (short term), -20°C (long…

ME0328

ME0328Band: www.medchemexpress.comSelective Inhibitor of PARP-3CAS No:1445251-22-8 Chemical Name: ME-0328; 3,4-Dihydro-4-oxo-3,4-Dihydro-4-oxo-N--2-quinazolinepropanamide; 3-(4-Oxo-3,4-dihydro-quinazolin-2-yl)-N-(1-phenyl-ethyl)-propionamide MLN4928 Molecular Formula C19H19N3O2 Molecular Weight 321.4 CAS Numbers 1445251-22-8 Storage Condition 0°C (short term), -20°C (long term), desiccated Solubility…

GW501516

GW501516Band: www.medchemexpress.coma potent and selective peroxisome proliferator-activated receptor (PPAR) β/δ modulator.CAS No:317318-70-0 VX-769 Molecular Formula C21H18F3NO3S2 Molecular Weight 453.5 CAS Numbers 317318-70-0 Storage Condition 0°C (short term), -20°C (long term),…

WAY-169916

WAY-169916Band: www.medchemexpress.comNovel pathway-selective estrogen receptor (ER) inhibitor, inhibiting NF-kB transcriptional activity but being devoid of conventional estrogenic activityCAS No: 669764-18-5   Chemical Name: 4-(1-Allyl-7-(trifluoromethyl)-1H-indazol-3-yl)benzene-1,3-diol AMG 236 Molecular Formula C17H13F3N2O2 Molecular Weight 334.29…

VPC-14228

VPC-14228Band: www.medchemexpress.comNovel specific inhibitor of AR-DBD, inhibitimg both Y594A and Q592A mutants, blocking the interaction of the AR with androgen response elements in the nucleus.CAS No: 19983-28-9   Chemical Name: 4-(4-Phenylthiazol-2-yl)morpholine Reparixin…

U-18666A

U-18666ABand: www.medchemexpress.comInhibitor of cholesterol synthesis, inhibiting desmosterol Δ24-reductaseCAS No:3039-71-2 Chemical Name: NSC-70801; (3β)-3-androst-5-en-17-one hydrochloride; (3S,8R,9S,10R,13S,14S)-3--10,13-dimethyl-1,2,3,4,7,8,9,11,12,14,15,16-dodecahydrocyclopentaphenanthren-17-one hydrochloride LY2109765 Molecular Formula C25H41NO2 • HCl Molecular Weight 424.1 CAS Numbers 3039-71-2 Storage Condition 0°C…

TAK-013

TAK-013Band: www.medchemexpress.comNovel nonpeptide gonadotropin-releasing hormone antagonist CAS No: 308831-61-0   Chemical Name: Sufugolix; 1-methyl]-1--2,4-dioxo-3-phenylthienopyrimidin-6-yl]phenyl]-3-methoxyurea Pexidartinib Molecular Formula C36H31F2N5O4S Molecular Weight 667.7 CAS Numbers 308831-61-0 Storage Condition 0°C (short term), -20°C (long term),…

STX-64

STX-64Band: www.medchemexpress.comA potent, irreversible inhibitor of steroid sulfatase.CAS No:288628-05-7 Asunaprevir Molecular Formula C14H15NO5S Molecular Weight 309.34 CAS Numbers 288628-05-7 Storage Condition 0°C (short term), -20°C (long term), desiccated Solubility DMSO…

RI-2

RI-2Band: www.medchemexpress.comInhibitor of RAD51, specifically inhibiting homologous recombination (HR) repair in human cellsCAS No: 1417162-36-7   Chemical Name: RI2; 1-(3,4-Dichlorophenyl)-3-(4-methoxyphenyl)-4-morpholino-1H-pyrrole-2,5-dione OTX-019 Molecular Formula C21H18Cl2N2O4 Molecular Weight 433.28 CAS Numbers 1417162-36-7 Storage Condition…