Sat. Jul 27th, 2024

FQI1

FQI1Band: www.medchemexpress.comAntiproliferative inhibitor of transcription factor LSF (Late SV40 factor)CAS No: 599151-35-6 Chemical Name: 8-(2-Ethoxyphenyl)-7,8-dihydro-1,3-dioxoloquinolin-6(5H)-one; factor quinolinone inhibitor 1 Firategrast Molecular Formula C18H17NO4 Molecular Weight 311.33 CAS Numbers 599151-35-6 References…

Dafadine-A

Dafadine-ABand: www.medchemexpress.comThe first identified chemical inhibitor of DAF-9CAS No: 1065506-69-5 Chemical Name: 4--3-isoxazolyl}carbonyl)-4-piperidinyl]-pyridine SCH772985 Molecular Formula C23H25N3O3 Molecular Weight 391.46 CAS Numbers 1065506-69-5 References PubMed ID::http://www.ncbi.nlm.nih.gov/pubmed/18499566

CID-5951923

CID-5951923Band: www.medchemexpress.comKruppel-like factor 5 (KLF5) expression inhibitorCAS No: 749872-43-3 Chemical Name: 3-(3-Nitro-phenyl)-acrylic acid -methyl ester CUDC-908 Molecular Formula C16H18N2O7S Molecular Weight 382.39 CAS Numbers 749872-43-3 References PubMed ID::http://www.ncbi.nlm.nih.gov/pubmed/18499565

CCG-1423

CCG-1423Band: www.medchemexpress.comSelective inhibitor of Rho pathway-mediated signaling and activation of serum response factor (SRF) transcriptionCAS No: 285986-88-1  Chemical Name: N-​-​1-​methyl-​2-​oxoethoxy]-​3,​5-​bis(trifluoromethyl)-​benzamide Vanoxerine Molecular Formula C18H13ClF6N2O3 Molecular Weight 454.75 CAS Numbers 285986-88-1 References PubMed…

BRD32048

BRD32048Band: www.medchemexpress.comNovel inhibitor of the ETV1 transcription factor oncoproteinCAS No: 433694-46-3   Chemical Name: N-(4-Methoxy-phenyl)-6-piperidin-1-ylmethyl-triazine-2,4-diamine UNC0643 Molecular Formula C16H22N6O Molecular Weight 314.39 CAS Numbers 433694-46-3 References PubMed ID::http://www.ncbi.nlm.nih.gov/pubmed/18499565

Necrostatin-2 racemate (7-Cl-O-Nec1)

Necrostatin-2 racemate (7-Cl-O-Nec1)Band: www.medchemexpress.comPotent necroptosis inhibitor CAS No: 852391-15-2   Chemical Name: rac-Necrostatin-2; 5--3-methylimidazolidine-2,4-dione GS-9621 Molecular Formula C₁₃H₁₂ClN₃O₂ Molecular Weight 277.71 CAS Numbers 852391-15-2 Storage Condition 0°C (short term), -20°C (long term),…

Lenalidomide

LenalidomideBand: www.medchemexpress.comThalidomide analog known to display TNF-α secretion inhibition and possesses immunomodulatory properties CAS No:191732-72-6 Chemical Name: Revlimid; Revimid; CC-5013; (3S)-3-(4-Amino-1-oxo-1,3-dihydro-2H-isoindol-2-yl)piperidine-2,6-dione AZD2015 Molecular Formula C13H13N3O3 Molecular Weight 259.3 CAS Numbers 191732-72-6…

JTE-607 dihydrochloride

JTE-607 dihydrochlorideBand: www.medchemexpress.comCytokine release inhibitor, inhibiting production of IL-1ß, IL-8, IL-6, IL-10 and TNFalphaCAS No: 188791-09-5   Chemical Name: N-benzoyl]-L-phenylalanine ethyl ester dihydrochloride BI 2537 Molecular Formula C25H31Cl2N3O5 2HCl Molecular Weight 597.36…

GW788388

GW788388Band: www.medchemexpress.comPotent and selective inhibitor of TGF-beta type I receptor CAS No:452342-67-5 Chemical Name: 4-{4--pyridin-2-yl}-N-(tetrahydro-2H-pyran-4-yl)benzamide ACY-1216 Molecular Formula C₂₅H₂₃N₅O₂ Molecular Weight 425.48 CAS Numbers 452342-67-5 Storage Condition 0°C (short term), -20°C…

EVP4593 (CAY10470)

EVP4593 (CAY10470)Band: www.medchemexpress.comPotent inhibitor of NF-κB activation and TNFα production CAS No: 545380-34-5   Chemical Name: QNZ; N4-​-​4,​6-​quinazolinediamine; CAY10470 Ko 144 Molecular Formula C22H20N4O Molecular Weight 356.42 CAS Numbers 545380-34-5 Storage Condition…