Wed. Jul 23rd, 2025

JNJ-17203212

JNJ-17203212Band: www.medchemexpress.comPotent TRPV1 (VR1) vanilloid receptor antagonist  CAS No: 821768-06-3 Chemical Name: 4-(3-Trifluoromethylpyridin-2-yl)piperazine-1-carboxylic acid (5-trifluoromethylpyridin-2-yl)amide; JNJ17203212 AZD3966 Molecular Formula C17H15F6N5O Molecular Weight 419.32 CAS Numbers 821768-06-3 References PubMed ID::http://www.ncbi.nlm.nih.gov/pubmed/18497261

GSK2193874

GSK2193874Band: www.medchemexpress.comSelective and orally active blocker of transient receptor potential vanilloid 4 (TRPV4)CAS No: 1336960-13-4   Chemical Name: 3-(-1-ylmethyl)-7-bromo-N-(1-phenylcyclopropyl)-2--4-quinolinecarboxami NVP-BGJ399 Molecular Formula C37H38BrF3N4O Molecular Weight 691.62 CAS Numbers 1336960-13-4 Storage Condition 0°C…

GSK205

GSK205Band: www.medchemexpress.comSelective Transient receptor potential vanilloid 4 (TRPV4) antagonistCAS No: 1263130-79-5   Chemical Name: N-​​ethyl]​phenyl]​-​5-​(3-​pyridinyl)​-2-​thiazolamine  PF-04449914 Molecular Formula C24H24N4S Molecular Weight 400.54 CAS Numbers 1263130-79-5 Storage Condition 0°C (short term), -20°C (long…

AMG-9810

AMG-9810Band: www.medchemexpress.comA potent non-vanilloid antagonist of the TRPV1 receptor CAS No: 545395-94-6   Chemical Name: 2E-N-(2,3-Dihydro-1,4-benzodioxin-6-yl)-3--2-Propenamide 4-Deazaneplanocin A (hydrochloride) Molecular Formula C21H23NO3 Molecular Weight 337.4 CAS Numbers 545395-94-6 Storage Condition 0°C (short…

Vorapaxar Sulfate (SCH 530348)

Vorapaxar Sulfate (SCH 530348)Band: www.medchemexpress.comA thrombin receptor (PAR-1) antagonist for the prevention and treatment of atherothrombosis.CAS No:705260-08-8 Vatalanib Molecular Formula C29H35FN2O8S Molecular Weight 590.66 CAS Numbers 705260-08-8 Storage Condition 0°C…

S1RA HCl

S1RA HClBand: www.medchemexpress.com A potent and selective sigma-1 receptorCAS No:1265917-14-3 Necrosulfonamide Molecular Formula C20H24ClN3O2 Molecular Weight 373.88 CAS Numbers 1265917-14-3 Storage Condition 0°C (short term), -20°C (long term), desiccated Solubility DMSO…

NE100 Hydrochloride

NE100 HydrochlorideBand: www.medchemexpress.comPotent and selective Sigma-1 receptor antagonist CAS No: 149409-57-4   Chemical Name: 4-Methoxy-3-(2-phenylethoxy)-N,Ndipropylbenzeneethanamine Hydrochloride Tonabersat Molecular Formula C23H34ClNO2 Molecular Weight 391.97 CAS Numbers 149409-57-4 Storage Condition 0°C (short term), -20°C…

Naloxonazine Dihydrochloride

Naloxonazine DihydrochlorideBand: www.medchemexpress.comPotent opioid antagonist, selective for μ1 receptors.CAS No:880759-65-9 Chemical Name: Bis- hydrazine dihydrochloride 1-NM-PP2 Molecular Formula C38H42N4O6.2HCl Molecular Weight 723.69 CAS Numbers 880759-65-9 Storage Condition 0°C (short term), -20°C (long term),…

ML138

ML138Band: www.medchemexpress.comSelective agonist of kappa opioid receptors (KOR)CAS No: 1355243-24-1 Chemical Name: 2--4-(furan-2-ylmethyl)-1,2,4-triazol-3-yl]pyridine; ML138; CID-44601470 CX-5462 Molecular Formula C19H14Cl2N4OS Molecular Weight 417.31 CAS Numbers 1355243-24-1 References PubMed ID::http://www.ncbi.nlm.nih.gov/pubmed/18496845

BW373U86 dihydrobromide

BW373U86 dihydrobromideBand: www.medchemexpress.comPotent, non-peptide delta-opioid receptor agonist. LDN193190 Molecular Formula C27H39Br2N3O2 Molecular Weight 597.43 CAS Numbers 1174661-92-7 Storage Condition 0°C (short term), -20°C (long term), desiccated Solubility DMSO Purity 98%…