Cytosporone BBand: www.medchemexpress.comThe first naturally occurring agonist for nuclear orphan receptor Nur77CAS No: 321661-62-5 Chemical Name: 3,5-Dihydroxy-2-(1-oxooctyl)benzeneacetic acid ethyl ester, Csn-B BMS 777608 Molecular Formula C18H26O5 Molecular Weight 322.40 CAS Numbers…
CarfilzomibBand: www.medchemexpress.comAn inhibitor the chymotrypsin-like activity of the 20S proteasomeCAS No:868540-17-4 Chemical Name:PR-171 CB-5084 Molecular Formula C40H57N5O7 Molecular Weight 719.91 CAS Numbers 868540-17-4 Storage Condition 0°C (short term), -20°C (long…
BMS-453Band: www.medchemexpress.comRetinoic acid receptor (RAR) antagonist and potent testicular toxinCAS No: 166977-43-1 Chemical Name: 4--benzoic acid Mdivi-2 Molecular Formula C27H24O2 Molecular Weight 380.48 CAS Numbers 166977-43-1 References PubMed ID：:http://www.ncbi.nlm.nih.gov/pubmed/18497713
KDM4B-IN-B3Band: www.medchemexpress.comNovel KDM4 inhibitor, blocking the binding of KDM4B to the PLK1 promoter, suppressing the expression of AR and BMYB-regulated genes Chemical Name: KDM4B Inhibitor B3; 3-(8-Hydroxyquinolin-6-yl)-N-(3-phenylpropyl)benzamide; NCGC00244536 Tebipenem Molecular Formula…
BarbadinBand: www.medchemexpress.comNovel selective β-arrestin/β2-adaptin inhibitor, blocking agonist-promoted endocytosis of the prototypical β2-adrenergic (β2AR), V2-vasopressin (V2R) and angiotensin-II type-1 (AT1R) receptors, showing no affectinng on β-arrestin-independent (transferrin) or AP2-independent (endothelin-A) receptor…
CMF-019 PotassiumBand: www.medchemexpress.comThe first potent biased small molecule agonist at the apelin receptor, increasing cardiac contractility in vivoCAS No: 1993426-69-9 Chemical Name: Potassium 3(S)-{-amino}-5-methyl-hexanoate LCL162 Molecular Formula C25H32KN3O3S Molecular Weight 493.70…
CMF-019Band: www.medchemexpress.comThe first potent biased small molecule agonist at the apelin receptor, increasing cardiac contractility in vivoCAS No: 1586787-08-7 Chemical Name: 3(S)-{-amino}-5-methyl-hexanoate TGR-1203 Molecular Formula C25H33N3O3S Molecular Weight 454.60 CAS…
MRT-10Band: www.medchemexpress.comSmoothened (Smo) receptor antagonistCAS No:330829-30-6 Chemical Name: N-amino]thioxomethyl]-3,4,5-trimethoxybenzamide Losmapimod Molecular Formula C24H23N3O5S Molecular Weight 465.52 CAS Numbers 330829-30-6 Storage Condition 0°C (short term), -20°C (long term), desiccated Solubility DMSO Purity…
Rilmenidine hemifumarateBand: www.medchemexpress.comSelective I1 imidazoline receptor agonistCAS No: 207572-68-7 Chemical Name: Oxaminozoline hemifumarate; N-(Dicyclopropylmethyl)-4,5-dihydro-2-oxazolamine hemifumarate salt Paritaprevir Molecular Formula C12H13N2O3 Molecular Weight 238.28 CAS Numbers 207572-68-7 Storage Condition 0°C (short term), -20°C…
ML314Band: www.medchemexpress.comNovel agonist of Neurotesin 1 Receptor (NTR1)CAS No: 1448895-09-7 Chemical Name: 2-Cyclopropyl-6,7-dimethoxy-4-quinazoline THZ2 Molecular Formula C22H26Cl2N2O9 Molecular Weight 421.36 CAS Numbers 858474-14-3 References PubMed ID：:http://www.ncbi.nlm.nih.gov/pubmed/18497484