Sat. Aug 16th, 2025

ML233

ML233Band: www.medchemexpress.comFunctional Agonist of the Apelin (APJ) ReceptorCAS No:1776055-05-0 Chemical Name: (E)-2-cyclohexyl-5-methyl-4-(phenylsulfonyloxyimino)cyclohexa-2,5-dienone; CID-46905036 Quisinostat Molecular Formula C19H21NO4S Molecular Weight 359.44 CAS Numbers 1776055-05-0 Storage Condition 0°C (short term), -20°C (long…

ML221

ML221Band: www.medchemexpress.comFunctional antagonist of the apelin (APJ) receptorCAS No: 877636-42-5 Chemical Name: -4-nitrobenzoate; CID-7217941 CH5424810 Molecular Formula C17H11N3O6S Molecular Weight 385.35 CAS Numbers 877636-42-5 Storage Condition 0°C (short term), -20°C…

ML194

ML194Band: www.medchemexpress.comGPR35 antagonistCAS No: 264233-05-8 Selumetinib Molecular Formula C17H19F2N5O2S Molecular Weight 395.43 Storage Condition -20C Solubility DMSO: soluble15 mg/mL References PubMed ID::http://www.ncbi.nlm.nih.gov/pubmed/18556747

ML 00253764 hydrochloride

ML 00253764 hydrochlorideBand: www.medchemexpress.comNon-peptide, melanocortin MC4 receptor antagonist (IC50 values are 0.32, 0.81 and 2.12 μM for MC4, MC3 and MC5 receptors respectively). Decreases cAMP accumulation in HEK-293 cells expressing…

LY-2157299

LY-2157299Band: www.medchemexpress.comPotent TGFβ receptor I (TβRI) inhibitor CAS No:700874-72-2 Dinaciclib Molecular Formula C22H19N5O Molecular Weight 369.42 CAS Numbers 700874-72-2 Storage Condition 0°C (short term), -20°C (long term), desiccated Solubility DMSO Purity…

JYL1421

JYL1421Band: www.medchemexpress.comSelective TRPV1 receptor antagonistCAS No: 401907-26-4   Chemical Name: N-(4-carbonothioyl)amino)methyl]-2-fluorophenyl)                               methanesulfonamide; SC0030 AZD-7770 Molecular Formula C20H26FN3O2S2 Molecular Weight 423.57 CAS Numbers 401907-26-4 Storage Condition 4C Solubility DMSO References PubMed ID::http://www.ncbi.nlm.nih.gov/pubmed/18556629

JTE-013

JTE-013Band: www.medchemexpress.comSphingosine 1-phosphate (S1P) receptor antagonistCAS No: 383150-41-2   Chemical Name: 1-pyridin-6-yl]-4-(2,6-dichloro-                               4-pyridinyl)-semicarbazide BAY 41-2280 Molecular Formula C17H19Cl2N7O Molecular Weight 408.29 CAS Numbers 383150-41-2 References PubMed ID::http://www.ncbi.nlm.nih.gov/pubmed/18556627

INT-747 (Obeticholic acid)

INT-747 (Obeticholic acid)Band: www.medchemexpress.comA potent and selective FXR agonist(EC50=99 nM) endowed with anticholestatic activity.CAS No:459789-99-2 BMS 777615 Molecular Formula C26H44O4 Molecular Weight 420.63 CAS Numbers 459789-99-2 Storage Condition 0°C (short…

Icilin

IcilinBand: www.medchemexpress.comNovel activator of the cold receptors TRPM8 (CMR1) and TRPA1 (ANKTM1/TRPN1) CAS No:36945-98-9 Chemical Name: 1-(2-Hydroxyphenyl)-4-(3-nitrophenyl)-1,2,3,6-tetra­hydro­pyrimidin-2-one, AG-3-5 CB-5091 Molecular Formula C16H13N3O4 Molecular Weight 311.3 CAS Numbers 36945-98-9 Storage Condition 0°C…

HJC0197

HJC0197Band: www.medchemexpress.comNovel Epac antagonistCAS No: 1383539-73-8   Chemical Name: 4-Cyclopentyl-2-(2,5-dimethylbenzylsulfanyl)-6-oxo-1,6-dihydropyrimidine-5-carbonitrile Mdivi-9 Molecular Formula C19H21N3OS Molecular Weight 339.45 CAS Numbers 1383539-73-8 Storage Condition 0°C (short term), -20°C (long term), desiccated Solubility DMSO Purity…